A Regioselective Synthesis of E-Guggulsterone
نویسندگان
چکیده
We have successfully prepared E-guggulsterone from 16,17-epoxypregnenolone in 84% yield over two steps via a hydrazine reduction and Oppenhauer oxidation. Additionally, isomerization was induced by heat, light (hν) and acid catalysis to convert Eguggulsterone into the corresponding Z isomer.
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